GLP-1 / Metabolic

Tirzepatide

FDA approved

Also known as: Mounjaro, Zepbound

The first dual incretin — superior to GLP-1 alone on weight, glucose, and metabolic markers.

Mechanism

GLP-1 / GIP dual agonist. The first dual incretin — superior to GLP-1 alone on weight, glucose, and metabolic markers. For full mechanism, dosing protocol, and stacking guidance, ask the AI Advisor or open the compound in-app.

Peer-Reviewed Studies (3)

Tirzepatide Once Weekly for Obesity (SURMOUNT-1)

NEJM · 2022

22.5% mean weight loss at 72 weeks; 36.2% lost ≥25%.

PubMed PMID 35658024

Tirzepatide vs Semaglutide in T2D (SURPASS-2)

NEJM · 2021

Superior HbA1c reduction (-2.0% to -2.3%) and weight loss.

PubMed PMID 34170647

Tirzepatide for HFpEF and Obesity (SUMMIT)

NEJM · 2024

Improved HFpEF symptoms and exercise capacity.

PubMed PMID 39555827

Related Compounds